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2022
N. C. Desai, Bhatt, K., Jadeja, D. J., Mehta, H. K., Khedkar, V. M., and Sarkar, D., β€œConventional and microwave-assisted organic synthesis of novel antimycobacterial agents bearing furan and pyridine hybrids”, Drug Development Research, vol. 83, no. 2, pp. 416-431, 2022.
D. D. Subhedar, Shaikh, M. H., Nagargoje, A. A., Sarkar, D., Khedkar, V. M., and Shingate, B. B., β€œ[DBUH][OAc]-catalyzed domino synthesis of novel benzimidazole incorporated 3,5-Bis (Arylidene)-4-piperidones as potential antitubercular agents”, Polycyclic Aromatic Compounds, vol. 42, no. 10, pp. 7010-7024, 2022.
P. S. Bhale, V. Chavan, H., Shringare, S. N., Khedkar, V. M., Tigote, R. M., Mali, N. N., Jadhav, T. D., Kamble, N. B., Kolat, S. P., Bandgar, B. P., and Patil, H. S., β€œDesign, synthesis of anticancer and anti-inflammatory 4-(1-methyl-1H-indol-3-yl)-6-(methylthio) pyrimidine-5-carbonitriles”, Synthetic Communications, vol. 52, no. 5, pp. 733-744, 2022.
M. H. Shaikh, Subhedar, D. D., Akolkar, S. V., Nagargoje, A. A., Khedkar, V. M., Sarkar, D., and Shingate, B. B., β€œTetrazoloquinoline-1,2,3-triazole derivatives as antimicrobial agents: synthesis, biological evaluation and molecular docking study”, Polycyclic Aromatic Compounds, vol. 42, no. 4, pp. 1920-1941, 2022.
V. S. Honmore, Natu, A. D., Khedkar, V. M., Arkile, M. A., Sarkar, D., and Rojatkar, S. R., β€œTwo antibacterial spiro compounds from the roots of Artemisia pallens wall: evidence from molecular docking”, Natural Product Research, vol. 36, no. 10, pp. 2465-2472, 2022.
2021
T. S. Chitre, Asgaonkar, K. D., Vikhe, A. B., Patil, S. M., Garud, D. R., Khedkar, V. M., Sarkar, D., Nawale, L. U., and Yeware, A., β€œIn silico studies, synthesis and antitubercular activity of some novel quinoline - azitidinone derivatives”, Current Computer-Aided Drug Design, vol. 17, no. 1, pp. 134-143, 2021.
A. B. Danne, ,, Sangshetti, J. N., Khedkar, V. M., and Shingate, B. B., β€œNew 1,2,3-triazole-appended bis-pyrazoles: synthesis, bioevaluation, and molecular docking”, ACS Omega, vol. 6, no. 38, pp. 24879-24890, 2021.
2020
B. B. Kashid, Salunkhe, P. H., Dongare, B. B., More, K. R., Khedkar, V. M., and Ghanwat, A. A., β€œSynthesis of novel of 2, 5-disubstituted 1, 3, 4-oxadiazole derivatives and their in vitro anti-inflammatory, anti-oxidant evaluation, and molecular docking study”, Bioorganic & Medicinal Chemistry Letters, vol. 30, no. 12, p. 127136, 2020.
2019
A. Atmaram Upare, Gadekar, P. K., Sivaramakrishnan, H., Naik, N., Khedkar, V. M., Sarkar, D., Choudhari, A., and S. Roopan, M., β€œDesign, synthesis and biological evaluation of (E)-5-styryl-1,2,4-oxadiazoles as anti-tubercular agents”, Bioorganic Chemistry, vol. 86, pp. 507-512, 2019.
T. S. Chitre, Patil, S. M., Sujalegaonkar, A. G., Asgaonkar, K. D., Khedkar, V. M., Garud, D. R., Jha, P. C., Gaikwad, S. Y., Kulkarni, S., Choudhari, A., and Sarkar, D., β€œNon nucleoside reverse transcriptase inhibitors, molecular docking studies and antitubercular activity of thiazolidin-4-one derivatives”, Current Computer-Aided Drug Design, vol. 15, no. 5, pp. 433-444, 2019.
2018
D. D. Subhedar, Shaikh, M. H., Tupe, S. G., Deshpande, M. V., Khedkar, V. M., Jha, P. C., and Shingate, B. B., β€œFacile and solvent-free domino synthesis of new quinolidinyl-2,4-thiazolidinones: antifungal activityand molecular docking”, Mini-Reviews in Medicinal Chemistry, vol. 18, no. 7, pp. 622-630, 2018.
N. C. Desai, β€œSynthesis, biological evaluation, and molecular docking study of pyridine clubbed 1,3,4-oxadiazoles as potential antituberculars”, Synthetic Communications, vol. 48, no. 5, pp. 524-540, 2018.
A. B. Danne, Choudhari, A. S., Chakraborty, S., Sarkar, D., Khedkar, V. M., and Shingate, B. B., β€œTriazole-diindolylmethane conjugates as new antitubercular agents: synthesis, bioevaluation, and molecular docking”, MedChemComm, vol. 9, no. 7, pp. 1114-1130, 2018.
2017
M. B. Bhalerao, Dhumal, S. T., Deshmukh, A. R., Nawale, L. U., Khedkar, V. M., Sarkar, D., and Mane, R. A., β€œNew bithiazolyl hydrazones: novel synthesis, characterization and antitubercular evaluation”, Bioorganic & Medicinal Chemistry Letters, vol. 27, no. 2, pp. 288–294, 2017.
D. D. Subhedar, Shaikh, M. H., Nawale, L. U., Sarkar, D., Khedkar, V. M., and Shingate, B. B., β€œQuinolidene based monocarbonyl curcumin analogues as promising antimycobacterial agents: synthesis and molecular docking study”, Bioorganic & medicinal chemistry letters, vol. 27, no. 4, pp. 922-928, 2017.
D. D. Subhedar, Shaikh, M. H., Shingate, B. B., Nawale, L., Sarkar, D., Khedkar, V. M., Khan, F. A. Kalam, and Sangshetti, J. N., β€œQuinolidene-rhodanine conjugates: facile synthesis and biological evaluation”, European Journal of Medicinal Chemistry, vol. 125, pp. 385–399, 2017.
J. M. Divse, Mhaske, S. B., Charolkar, C. R., Sant, D. G., Tupe, S. G., Deshpande, M. V., Khedkar, V. M., Nawale, L. U., Sarkar, D., and Pore, V. S., β€œSynthesis and biological evaluation of new fluconazole Ξ²-lactam conjugates linked via 1,2,3-triazole”, New Journal of Chemistry, vol. 41, no. 2, pp. 470-479, 2017.
N. D. Rode, Sonawane, A. D., Nawale, L., Khedkar, V. M., Joshi, R. A., Likhite, A. P., Sarkar, D., and Joshi, R. R., β€œSynthesis, biological evaluation, and molecular docking studies of novel 3-aryl-5-(alkyl-thio)-1H-1,2,4-triazoles derivatives targeting Mycobacterium tuberculosis”, Chemical Biology & Drug Design, vol. 90, no. 6, pp. 1206-1214, 2017.
V. E. Goud, Sivaramakrishna, A., Vijayakrishna, K., Rao, C. V. S. Brah, Khedkar, V. M., and Jha, P. C., β€œSynthesis, structure and DNA interaction studies of bisphosphoramides: theoretical and experimental insights”, Inorganica Chimica Acta, vol. 461, pp. 84-91, 2017.
2016
P. K. Gadekar, Roychowdhury, A., Kharkar, P. S., Khedkar, V. M., Arkile, M. A., Manek, H., Sarkar, D., Sharma, R., Vijayakumar, V., and Sarveswari, S., β€œDesign, synthesis and biological evaluation of novel azaspiro analogs of linezolid as antibacterial and antitubercular agents”, European Journal of Medicinal Chemistry, vol. 122, pp. 475-487, 2016.
N. C. Desai, Kotadiya, G. M., Trivedi, A. R., Khedkar, V. M., and Jha, P. C., β€œDesign, synthesis, and biological evaluation of novel fluorinated pyrazole encompassing pyridyl 1,3,4-oxadiazole motifs”, Medicinal Chemistry Research, vol. 25, no. 11, pp. 2698-2717, 2016.
D. D. Subhedar, Shaikh, M. H., Khan, F. A. Kalam, Sangshetti, J. N., Khedkar, V. M., and Shingate, B. B., β€œFacile synthesis of new N-sulfonamidyl-4-thiazolidinone derivatives and their biological evaluation”, New Journal of Chemistry, vol. 40, no. 4, pp. 3047-3058, 2016.
V. S. Honmore, Rojatkar, S. R., Nawale, L. U., Arkile, M. A., Khedkar, V. M., Natu, A. D., and Sarkar, D., β€œIn vitro and ex vivo antitubercular activity of diarylheptanoids from the rhizomes of alpinia officinarum hance”, Natural Product Research, vol. 30, no. 24, pp. 2825-2830, 2016.
V. S. Honmore, Kandhare, A. D., Kadam, P. P., Khedkar, V. M., Sarkar, D., Bodhankar, S. L., Zanwar, A. A., Rojatkar, S. R., and Natu, A. D., β€œIsolates of alpinia officinarum hance as COX-2 inhibitors: evidence from anti-inflammatory, antioxidant and molecular docking studies”, International Immunopharmacology, vol. 33, pp. 8-17, 2016.
S. K. Patel, Khedkar, V. M., Jha, P. C., Jasrai, Y. T., Pandya, H. A., George, L. - B., Highland, H. N., and Skelton, A. A., β€œMolecular interaction of selected phytochemicals under the charged environment of Plasmodium falciparum chloroquine resistance transporter (PfCRT) model”, Journal of Biomolecular Structure & Dynamics, vol. 34, no. 2, pp. 290-303, 2016.
R. R. Kulkarni, Shurpali, K., Khedkar, V. M., Puranik, V. G., Sarkar, D., and Joshi, S. P., β€œNew pimarane diterpenes and other antimycobacterial metabolites from anisochilus verticillatus”, Natural Product Research, vol. 30, no. 6, pp. 675-681, 2016.
D. D. Subhedar, Shaikh, M. H., Shingate, B. B., Nawale, L., Sarkar, D., and Khedkar, V. M., β€œNovel tetrazoloquinoline-thiazolidinone conjugates as possible antitubercular agents: synthesis and molecular docking”, Medchemcomm, vol. 7, no. 9, pp. 1832-1848, 2016.
S. T. Dhumal, Deshmukh, A. R., Bhosle, M. R., Khedkar, V. M., Nawale, L. U., Sarkar, D., and Mane, R. A., β€œSynthesis and antitubercular activity of new 1,3,4-oxadiazoles bearing pyridyl and thiazolyl scaffolds”, Bioorganic & Medicinal Chemistry Letters, vol. 26, no. 15, pp. 3646-3651, 2016.
P. S. Mahajan, Nikam, M. D., Nawale, L. U., Khedkar, V. M., Sarkar, D., and Gill, C. H., β€œSynthesis and antitubercular activity of new benzo[b]thiophenes”, ACS Medicinal Chemistry Letters, vol. 7, no. 8, pp. 751-756, 2016.
M. H. Shaikh, Subhedar, D. D., Arkile, M. A., Khedkar, V. M., Jadhav, N. J., Sarkar, D., and Shingate, B. B., β€œSynthesis and bioactivity of novel triazole incorporated benzothiazinone derivatives as antitubercular and antioxidant agent”, Bioorganic & Medicinal Chemistry Letters, vol. 26, no. 2, pp. 561-569, 2016.
T. S. Chitre, Asgaonkar, K. D., Miniyar, P. B., Dharme, A. B., Arkile, M. A., Yeware, A., Sarkar, D., Khedkar, V. M., and Jha, P. C., β€œSynthesis and docking studies of pyrazine-thiazolidinone hybrid scaffold targeting dormant tuberculosis”, Bioorganic & Medicinal Chemistry Letters, vol. 26, no. 9, pp. 2224-2228, 2016.
M. H. Shaikh, Subhedar, D. D., Shingate, B. B., Khan, F. A. Kalam, Sangshetti, J. N., Khedkar, V. M., Nawale, L., Sarkar, D., Navale, G. R., and Shinde, S. S., β€œSynthesis, biological evaluation and molecular docking of novel coumarin incorporated triazoles as antitubercular, antioxidant and antimicrobial agents”, Medicinal Chemistry Research, vol. 25, no. 4, pp. 790-804, 2016.
P. S. Mahajan, Nikam, M. D., Khedkar, V. M., Jha, P. C., Sarkar, D., and Gill, C. H., β€œSynthesis, biological evaluation and molecular docking studies of N-acylheteroaryl hydrazone derivatives as antioxidant and anti-inflammatory agents”, Research on Chemical Intermediates, vol. 42, no. 3, pp. 2707-2729, 2016.
N. C. Desai, Somani, H., Trivedi, A., Bhatt, K., Nawale, L., Khedkar, V. M., Jha, P. C., and Sarkar, D., β€œSynthesis, biological evaluation and molecular docking study of some novel indole and pyridine based 1,3,4-oxadiazole derivatives as potential antitubercular agents”, Bioorganic & Medicinal Chemistry Letters, vol. 26, no. 7, pp. 1776-1783, 2016.
N. C. Desai, Kotadiya, G. M., Trivedi, A. R., Khedkar, V. M., and Jha, P. C., β€œSynthesis, biological valuation, and QSAR studies of novel pyrazole bearing pyridyl oxadiazole analogues as potential antimicrobial agents”, Medicinal Chemistry Research, vol. 25, no. 4, pp. 712-727, 2016.
2015
K. Manojkumar, Charan, K. T. Prabhu, Sivaramakrishna, A., Jha, P. C., Khedkar, V. M., Siva, R., Jayaraman, G., and Vijayakrishna, K., β€œBiophysical characterization and molecular docking studies of imidazolium based polyelectrolytes-DNA complexes: role of hydrophobicity”, Biomacromolecules, vol. 16, no. 3, pp. 894-903, 2015.
V. S. Pore, Divse, J. M., Charolkar, C. R., Nawale, L. U., Khedkar, V. M., and Sarkar, D., β€œDesign and synthesis of 11 alpha-substituted bile acid derivatives as potential anti-tuberculosis agents”, Bioorganic & Medicinal Chemistry Letters, vol. 25, no. 19, pp. 4185-4190, 2015.
K. T. Prabhu Charan, Ranjan, P., Manojkumar, K., Pothanagandhi, N., Jha, P. C., Khedkar, V. M., Sivaramakrishna, A., and Vijayakrishna, K., β€œEvaluation of imidazolium-based ionic liquids towards vermicidal activity: in vitro & in silico studies”, RSC Advances, vol. 5, no. 92, pp. 75415-75424, 2015.
R. R. Joshi, Barchha, A., Khedkar, V. M., Pissurlenkar, R. R. S., Sarkar, S., Sarkar, D., Joshi, R. R., Joshi, R. A., Shah, A. K., and Coutinho, E. C., β€œTargeting dormant tuberculosis bacilli: results for molecules with a novel pyrimidone scaffold”, Chemical Biology & Drug Design, vol. 85, no. 2, pp. 201-207, 2015.
2013
R. P. Samal, Khedkar, V. M., Pissurlenkar, R. R. S., Bwalya, A. Gono, Tasdemir, D., Joshi, R. A., Rajamohanan, P. R., Puranik, V. G., and Coutinho, E. C., β€œDesign, synthesis, structural characterization by IR, 1H, 13C, 15N, 2D-NMR, X-ray diffraction and evaluation of a new class of phenylaminoacetic acid benzylidene hydrazines as pfENR inhibitors”, Chemical Biology & Drug Design, vol. 81, no. 6, pp. 715-729, 2013.