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2019
, ,, Wadgaonkar, P. P., Tapase, S. R., Kodam, K. M., Choudhari, A., and Sarkar, D., Click chemistry based multicomponent approach in the synthesis of spirochromenocarbazole tethered 1,2,3-triazoles as potential anticancer agents, Bioorganic Chemistry, vol. 85, pp. 475-486, 2019.
S. B. Baravkar, Wagh, M. A., Nawale, L. U., Choudhari, A. S., Bhansali, S., Sarkar, D., and Sanjayan, G. J., Design and synthesis of 2-amino-thiophene-proline-conjugates and their anti-tubercular activity against mycobacterium tuberculosis H37Ra, ChemistrySelect, vol. 4, no. 9, pp. 2851-2857, 2019.
A. Atmaram Upare, Gadekar, P. K., Sivaramakrishnan, H., Naik, N., Khedkar, V. M., Sarkar, D., Choudhari, A., and S. Roopan, M., Design, synthesis and biological evaluation of (E)-5-styryl-1,2,4-oxadiazoles as anti-tubercular agents, Bioorganic Chemistry, vol. 86, pp. 507-512, 2019.
S. P. Gample, Agrawal, S., and Sarkar, D., Evidence of nitrite acting as a stable and robust inducer of non-cultivability in Mycobacterium tuberculosis with physiological relevance, Scientific Reports, vol. 9, p. 9261, 2019.
A. Yeware, Agrawal, S., and Sarkar, D., High content screening assay for identifying inhibitors against active and dormant state intracellular Mycobacterium tuberculosis, Journal of Microbiological Methods, vol. 164, 2019.
T. S. Chitre, Patil, S. M., Sujalegaonkar, A. G., Asgaonkar, K. D., Khedkar, V. M., Garud, D. R., Jha, P. C., Gaikwad, S. Y., Kulkarni, S., Choudhari, A., and Sarkar, D., Non nucleoside reverse transcriptase inhibitors, molecular docking studies and antitubercular activity of thiazolidin-4-one derivatives, Current Computer-Aided Drug Design, vol. 15, no. 5, pp. 433-444, 2019.
P. Miniyar, Mahajan, A., Anuse, D., Kumar, A., Barmade, M., Sarkar, D., Arkile, M., and Khedkar, V., Recursive partitioning analysis and anti-tubercular screening of 3-aminopyrazine-2-carbohydrazide derivatives, Letters in Drug Design & Discovery, vol. 16, no. 11, pp. 1264-1275, 2019.
V. Shinde, Mahulikar, P., Mhaske, P. C., Chakraborty, S., Choudhari, A., Phalle, S., Choudhari, P., and Sarkar, D., Synthesis and antimycobacterial evaluation of new 5-(1-benzyl-1H-1,2,3-triazol-4-yl)-4-methyl-2-arylthiazole derivatives, Medicinal Chemistry Research, vol. 28, no. 6, pp. 805-819, 2019.
U. B. Karale, Krishna, V. Siva, E. Krishna, V., Choudhari, A. S., Shukla, M., Gaikwad, V. R., Mahizhaveni, B., Chopra, S., Misra, S., Sarkar, D., Sriram, D., Dusthackeer, V. N. Azger, and Rode, H. B., Synthesis and biological evaluation of 2,4,5-trisubstituted thiazoles as antituberculosis agents effective against drug-resistant tuberculosis, European Journal of Medicinal Chemistry, vol. 178, pp. 315-328, 2019.
V. Shinde, Mhaske, P. C., Singh, A., Sarkar, D., and Mahulikar, P., Synthesis and biological evaluation of new 4-(4-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl)-2-phenylthiazole derivatives, Journal of Heterocyclic Chemistry, 2019.
A. P. Chavan, Deshpande, R. R., Borade, N. A., Shinde, A., Mhaske, P. C., Sarkar, D., and Bobade, V. D., Synthesis of new 1,3,4-oxadiazole and benzothiazolylthioether derivatives of 4-arylmethylidene-3-substituted-isoxazol-5(4H)-one as potential antimycobacterial agents, Medicinal Chemistry Research, vol. 28, no. 11, pp. 1873-1884, 2019.
S. J. Takate, Shinde, A. D., Karale, B. K., Akolkar, H., Nawale, L., Sarkar, D., and Mhaske, P. C., Thiazolyl-pyrazole derivatives as potential antimycobacterial agents, Bioorganic & Medicinal Chemistry Letters, vol. 29, no. 10, pp. 1199-1202, 2019.
A. Yeware, Gample, S., Agrawal, S., and Sarkar, D., Using diphenyleneiodonium to induce a viable but non-culturable phenotype in Mycobacterium tuberculosis and its metabolomics analysis, Plos One, vol. 14, no. 8, p. e0220628, 2019.
2021
R. Balasaheb Aher and Sarkar, D., 2D-QSAR modeling and two-fold classification of 1,2,4-triazole derivatives for antitubercular potency against the dormant stage of Mycobacterium tuberculosis, Molecular Diversity, vol. 26, no. 2, pp. 1227-1242, 2021.
T. S. Chitre, Asgaonkar, K. D., Vikhe, A. B., Patil, S. M., Garud, D. R., Khedkar, V. M., Sarkar, D., Nawale, L. U., and Yeware, A., In silico studies, synthesis and antitubercular activity of some novel quinoline - azitidinone derivatives, Current Computer-Aided Drug Design, vol. 17, no. 1, pp. 134-143, 2021.
V. Honmore, Kalyankar, V., Natu, A., Khedkar, V., Sarkar, D., and Rojatkar, S., In vitro antitubercular screening and in silico study of germacradienolide from blainvillea latifolia, Asian Journal of Chemistry, vol. 33, no. 12, pp. 3129-3133, 2021.
S. Agrawal, Gample, S., Yeware, A., and Sarkar, D., Novel gene similar to nitrite reductase (NO forming) plays potentially important role in the latency of tuberculosis, Scientific Reports, vol. 11, no. 1, p. 19813, 2021.
R. Balasaheb Aher and Sarkar, D., Online tools and antiviral databases for the development of drugs against coronaviruses, in In Silico Modeling of Drugs Against Coronaviruses: Computational Tools and Protocols, K. Roy, Ed. New York, NY: Springer US, 2021, pp. 717–734.
R. Balasaheb Aher and Sarkar, D., Pharmacophore modeling of pretomanid (PA-824) derivatives for antitubercular potency against replicating and non-replicating Mycobacterium tuberculosis, Journal of Biomolecular Structure & Dynamics, vol. 39, no. 3, pp. 889-900, 2021.
M. M. Pisal, Annadate, R. A., Athalye, M. C., Kumar, D., Chavan, S. P., Sarkar, D., and Borate, H. B., Synthesis and cell imaging applications of fluorescent mono/di/tri-heterocyclyl-2,6-dicyanoanilines (vol 27, pg 979, 2017), Bioorganic & Medicinal Chemistry Letters, vol. 32, p. 127737, 2021.
Y. K. Abhale, Shinde, A., Shelke, M., Nawale, L., Sarkar, D., and Mhaske, P. C., Synthesis of new 2-(thiazol-4-yl)thiazolidin-4-one derivatives as potential anti-mycobacterial agents, Bioorganic Chemistry, vol. 115, p. 105192, 2021.
2022
D. D. Subhedar, Shaikh, M. H., Nagargoje, A. A., V. Akolkar, S., Bhansali, S. G., Sarkar, D., and Shingate, B. B., Amide-linked monocarbonyl curcumin analogues: efficient synthesis, antitubercular activity and molecular docking study, Polycyclic Aromatic Compounds, vol. 45, no. 5, pp. 2655-2671, 2022.
N. C. Desai, Bhatt, K., Jadeja, D. J., Mehta, H. K., Khedkar, V. M., and Sarkar, D., Conventional and microwave-assisted organic synthesis of novel antimycobacterial agents bearing furan and pyridine hybrids, Drug Development Research, vol. 83, no. 2, pp. 416-431, 2022.
D. D. Subhedar, Shaikh, M. H., Nagargoje, A. A., Sarkar, D., Khedkar, V. M., and Shingate, B. B., [DBUH][OAc]-catalyzed domino synthesis of novel benzimidazole incorporated 3,5-Bis (Arylidene)-4-piperidones as potential antitubercular agents, Polycyclic Aromatic Compounds, vol. 42, no. 10, pp. 7010-7024, 2022.
S. Sarkar, Swami, S., Soni, S. Kumar, Holien, J. K., Khan, A., Korwar, A. M., Likhite, A. P., Joshi, R. A., Joshi, R. R., and Sarkar, D., Detection of a target protein (GroEl2) in Mycobacterium tuberculosis using a derivative of 1,2,4-triazolethiols, Molecular Diversity, vol. 26, no. 5, pp. 2535-2548, 2022.
G. Navale, Singh, S., Agrawal, S., Ghosh, C., Choudhury, A. Roy, Roy, P., Sarkar, D., and Ghosh, K., DNA binding, antitubercular, antibacterial and anticancer studies of newly designed piano-stool ruthenium(ii) complexes, Dalton Transactions, vol. 51, no. 42, pp. 16371-16382, 2022.
A. Yeware, Akhtar, S., and Sarkar, D., Probes and techniques used in active and the hypoxia-based dormant state of an antitubercular drug screening assay, Medicine in Drug Discovery, vol. 13, p. 100115, 2022.
J. L. Nalawade, Mhaske, P. C., Shinde, A. D., Chavan, A. P., Abhale, Y. K., Sarkar, D., and Bobade, V. D., Synthesis and antimycobacterial screening of a novel series of alpha-amino acids containing thiazole linker, ARKIVOC, 2022.
S. M. Jagadale, Abhale, Y. K., Pawar, H. R., Shinde, A., Bobade, V. D., Chavan, A. P., Sarkar, D., and Mhaske, P. C., Synthesis of new thiazole and pyrazole clubbed 1,2,3-triazol derivatives as potential antimycobacterial and antibacterial agents, Polycyclic Aromatic Compounds, vol. 42, no. 6, pp. 3216-3237, 2022.
M. H. Shaikh, Subhedar, D. D., Akolkar, S. V., Nagargoje, A. A., Khedkar, V. M., Sarkar, D., and Shingate, B. B., Tetrazoloquinoline-1,2,3-triazole derivatives as antimicrobial agents: synthesis, biological evaluation and molecular docking study, Polycyclic Aromatic Compounds, vol. 42, no. 4, pp. 1920-1941, 2022.
V. S. Honmore, Natu, A. D., Khedkar, V. M., Arkile, M. A., Sarkar, D., and Rojatkar, S. R., Two antibacterial spiro compounds from the roots of Artemisia pallens wall: evidence from molecular docking, Natural Product Research, vol. 36, no. 10, pp. 2465-2472, 2022.

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