TY - JOUR T1 - Hypervalent-iodine-mediated oxidation followed by the acetoxylation/tosylation of alpha-substituted benzylamines to obtain alpha-acyloxy/tosyloxy ketones JF - New Journal of Chemistry Y1 - 2022 A1 - Rupanawar, Bapurao D. A1 - Mane, Kishor D. A1 - Suryavanshi, Gurunath AB -

An efficient and metal-free method has been developed for the sequential oxidation of alpha-alkylbenzylamines followed by acetoxylation or tosylation for the synthesis of alpha-acyloxy/tosyloxy ketones using hypervalent iodine(iii). The employment of a simple starting material, broad substrate scope and operational simplicity are the key features of this protocol.

VL - 46 IS - 35 U3 -

Foreign

U4 -

3.925

ER -