@article {47427,
	title = {Short enantioselective total synthesis of (+)-tofacitinib},
	journal = {Tetrahedron Letters},
	volume = {67},
	year = {2021},
	month = {MAR},
	pages = {152838},
	type = {Article},
	abstract = {<p>An enantioselective total synthesis of Tofacitinib (CP-690,550), a Janus tyrosine kinase (JAK3) specific inhibitor has been achieved from the readily available 4-piperidone. Proline catalysed hydroxylation is the key step for the synthesis of enantiopure 1-benzyl-4-methylpiperidin-3-ol. (C) 2021 Elsevier Ltd. All rights reserved.</p>},
	keywords = {aminohydroxylation, Hydrogenation, L-proline, piperidone},
	issn = {0040-4039},
	doi = {10.1016/j.tetlet.2021.152838},
	author = {Mane, Kishor D. and Kamble, Rohit B. and Suryavanshi, Gurunath}
}
@article {48304,
	title = {Synthesis of 3 alkyl and 1,3-Bis(alkyl)indolizine amides from a-bromohydroxamates},
	journal = {Tetrahedron Letters},
	volume = {118},
	year = {2023},
	month = {MAR},
	pages = {154386},
	type = {Article},
	abstract = {<p>A simple and catalyst-free method has been developed for the synthesis of hindered indolizine amide derivatives from functionalized alkyl bromides. The reaction of a variety of indolizine derivatives with azaoxyallyl cations generated in situ from a-bromoamides afforded a wide range of synthetically important mono- and di-alkylated indolizine amide derivatives in good to excellent yields.@2023 Elsevier Ltd. All rights reserved.</p>
},
	keywords = {a -Bromohydroxamates, Amides, HFIP, Indolizine},
	issn = {0040-4039},
	doi = {10.1016/j.tetlet.2023.154386},
	author = {Mane, Kishor D. and Bagwe, Sagar S. and More, Satish G. and Suryavanshi, Gurunath}
}
